Setastine 59767-13-4
64294-95-7

Setastine (Loderix) is an antihistamine used to treat allergies and rhinitis.

Pharmacology

Pharmacodynamics

Setastine acts as a highly selective H₁ receptor antagonist. It has no anticholinergic, antiadrenergic, or antiserotonergic effects.

Pharmacokinetics

Setastine penetrates the blood-brain-barrier only weakly, hence, it is not sedating or is only mildly so.

read more [+]

Systematic (IUPAC) name:	1-[2-[1-(4-chlorophenyl)-1-phenyl-ethoxy]ethyl]azepane
Setastine CAS number:	59767-13-4 64294-95-7
ATC code:
PubChem:	43082
DrugBank:
Formula:
Molecular mass:	357.92 g/mol
Setastine Assay/Purity:	Typically NLT 98%

Products currently covered by valid US Patents are offered for R&D use in accordance with 35 USC 271(e)+A13(1). Any patent infringement and resulting liability is solely at buyer risk.