Pazinaclone 103255-66-9

Pazinaclone (DN-2327) is a sedative and anxiolytic drug in the cyclopyrrolone family of drugs. Other cyclopyrrolone drugs include zopiclone and eszopiclone. Pazinaclone has a very similar pharmacological profile to the benzodiazepine family of drugs including sedative and anxiolytic properties, but with less amnestic effects, and at low doses it is a relatively selective anxiolytic, with sedative effects only appearing at higher doses. Pazinaclone produces its sedative and anxiolytic effects by acting as a partial agonist at GABA_A benzodiazepine receptors, although pazinaclone is more subtype-selective than most benzodiazepines.

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Systematic (IUPAC) name:	2-(7-chloro-1,8-naphthyridin-2-yl)-3-[2-(1,4-dioxa-8- azaspiro[4.5]decan-8-yl)-2-oxoethyl]-3H-isoindol-1-one
Pazinaclone CAS number:	103255-66-9
ATC code:
PubChem:	59743
DrugBank:
Formula:	C25H23N4O4
Molecular mass:	478.928 g/mol
Pazinaclone Assay/Purity:	Typically NLT 98%

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